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Combined SFK/mTOR inhibition prevents rapamycin-induced feedback activation of AKT and elicits efficient tumor regression

Resistance to receptor tyrosine kinase (RTK) blockade in breast cancer is often mediated by activation of bypass pathways that sustain growth. Src and mammalian target of rapamycin (mTOR) are two intrinsic targets that are downstream of most RTKs. To date, limited clinical efficacy has been observed...

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Autors principals: Yori, Jennifer L., Lozada, Kristen L., Seachrist, Darcie D., Mosley, Jonathan D., Abdul-Karim, Fadi W., Booth, Christine N., Flask, Chris A., Keri, Ruth A.
Format: Artigo
Idioma:Inglês
Publicat: 2014
Matèries:
Accés en línia:https://ncbi.nlm.nih.gov/pmc/articles/PMC4155007/
https://ncbi.nlm.nih.gov/pubmed/25023728
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1158/0008-5472.CAN-13-3627
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