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Structure-based Ligand Design of Novel Human Toll-like Receptor 8 Agonists

Toll-like receptor (TLR)-8 agonists activate adaptive immune responses by inducing robust production of T helper 1-polarizing cytokines, suggesting that TLR8-active compounds may be promising candidate adjuvants. We recently reported pure TLR8 agonistic activity in a C2-butyl furo[2,3-c]quinoline. W...

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主要な著者: Kokatla, Hari Prasad, Sil, Diptesh, Tanji, Hiromi, Ohto, Umeharu, Malladi, Subbalakshmi S., Fox, Lauren M., Shimizu, Toshiyoki, David, Sunil A.
フォーマット: Artigo
言語:Inglês
出版事項: 2014
主題:
オンライン・アクセス:https://ncbi.nlm.nih.gov/pmc/articles/PMC4105021/
https://ncbi.nlm.nih.gov/pubmed/24474703
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1002/cmdc.201300573
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