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Chemically Accessible Hsp90 Inhibitor That Does Not Induce a Heat Shock Response

[Image: see text] Recent cancer therapies have focused on targeting biology networks through a single regulatory protein. Heat shock protein 90 (hsp90) is an ideal oncogenic target as it regulates over 400 client proteins and cochaperones. However, clinical inhibitors of hsp90 have had limited succe...

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Autores principales: Koay, Yen Chin, McConnell, Jeanette R., Wang, Yao, Kim, Seong Jong, Buckton, Laura K., Mansour, Flora, McAlpine, Shelli R.
Formato: Artigo
Lenguaje:Inglês
Publicado: American Chemical Society 2014
Acceso en línea:https://ncbi.nlm.nih.gov/pmc/articles/PMC4094262/
https://ncbi.nlm.nih.gov/pubmed/25050163
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/ml500114p
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