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Muscarinic acetylcholine receptor X-ray structures: potential implications for drug development

Muscarinic acetylcholine receptor antagonists are widely used as bronchodilating drugs in pulmonary medicine. The therapeutic efficacy of these agents depends on the blockade of M(3) muscarinic receptors expressed on airway smooth muscle cells. All muscarinic antagonists currently used as bronchodil...

Deskribapen osoa

Gorde:
Xehetasun bibliografikoak
Egile Nagusiak: Kruse, Andrew C., Hu, Jianxin, Kobilka, Brian K., Wess, Jürgen
Formatua: Artigo
Hizkuntza:Inglês
Argitaratua: 2014
Gaiak:
Sarrera elektronikoa:https://ncbi.nlm.nih.gov/pmc/articles/PMC4065632/
https://ncbi.nlm.nih.gov/pubmed/24662799
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1016/j.coph.2014.02.006
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