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Design, Synthesis, and Structure–Activity Relationships of Pyridoquinazolinecarboxamides as RNA Polymerase I Inhibitors

[Image: see text] RNA polymerase I (Pol I) is a dedicated polymerase that transcribes the 45S ribosomal (r) RNA precursor. The 45S rRNA precursor is subsequently processed into the mature 5.8S, 18S, and 28S rRNAs and assembled into ribosomes in the nucleolus. Pol I activity is commonly deregulated i...

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Dettagli Bibliografici
Autori principali: Colis, Laureen, Ernst, Glen, Sanders, Sara, Liu, Hester, Sirajuddin, Paul, Peltonen, Karita, DePasquale, Michael, Barrow, James C., Laiho, Marikki
Natura: Artigo
Lingua:Inglês
Pubblicazione: American Chemical Society 2014
Accesso online:https://ncbi.nlm.nih.gov/pmc/articles/PMC4059246/
https://ncbi.nlm.nih.gov/pubmed/24847734
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/jm5004842
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