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Conformational changes in dopamine transporter intracellular regions upon cocaine binding and dopamine translocation

The dopamine transporter (DAT), a member of the neurotransmitter:sodium symporter family, mediates the reuptake of dopamine at the synaptic cleft. DAT is the primary target for psychostimulants such as cocaine and amphetamine. We previously demonstrated that cocaine binding and dopamine transport al...

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Autors principals: Dehnes, Yvette, Shan, Jufang, Beuming, Thijs, Shi, Lei, Weinstein, Harel, Javitch, Jonathan A.
Format: Artigo
Idioma:Inglês
Publicat: 2014
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Accés en línia:https://ncbi.nlm.nih.gov/pmc/articles/PMC4058377/
https://ncbi.nlm.nih.gov/pubmed/24576496
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1016/j.neuint.2014.02.003
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