Wird geladen...

Effect of soluble epoxide hydrolase polymorphism on substrate and inhibitor selectivity and dimer formation

Epoxy FAs (EpFAs) are important lipid mediators that are mainly metabolized by soluble epoxide hydrolase (sEH). Thus, sEH inhibition is a promising therapeutic target to treat numerous ailments. Several sEH polymorphisms result in amino acid substitutions and alter enzyme activity. K55R and R287Q ar...

Ausführliche Beschreibung

Gespeichert in:
Bibliographische Detailangaben
Hauptverfasser: Morisseau, Christophe, Wecksler, Aaron T., Deng, Catherine, Dong, Hua, Yang, Jun, Lee, Kin Sing S., Kodani, Sean D., Hammock, Bruce D.
Format: Artigo
Sprache:Inglês
Veröffentlicht: The American Society for Biochemistry and Molecular Biology 2014
Schlagworte:
Online Zugang:https://ncbi.nlm.nih.gov/pmc/articles/PMC4031944/
https://ncbi.nlm.nih.gov/pubmed/24771868
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1194/jlr.M049718
Tags: Tag hinzufügen
Keine Tags, Fügen Sie den ersten Tag hinzu!