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Design and Potency of Dual Soluble Epoxide Hydrolase/Fatty Acid Amide Hydrolase Inhibitors

[Image: see text] Fatty acid amide hydrolase (FAAH) is responsible for regulating concentrations of the endocannabinoid arachidonoyl ethanolamide. Multiple FAAH inhibitors have been developed for clinical trials and have failed to demonstrate efficacy at treating pain, despite promising preclinical...

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Dettagli Bibliografici
Pubblicato in:ACS Omega
Autori principali: Kodani, Sean D., Wan, Debin, Wagner, Karen M., Hwang, Sung Hee, Morisseau, Christophe, Hammock, Bruce D.
Natura: Artigo
Lingua:Inglês
Pubblicazione: American Chemical Society 2018
Accesso online:https://ncbi.nlm.nih.gov/pmc/articles/PMC6210075/
https://ncbi.nlm.nih.gov/pubmed/30411058
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/acsomega.8b01625
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