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Evaluation of structural effects on 5-HT(2A) receptor antagonism by aporphines: identification of a new aporphine with 5-HT(2A) antagonist activity

A set of aporphine analogs related to nantenine was evaluated for antagonist activity at 5-HT(2A) and α(1A) adrenergic receptors. With regards to 5-HT(2A) receptor antagonism, a C2 allyl group is detrimental to activity. The chiral center of nantenine is not important for 5-HT(2A) antagonist activit...

पूर्ण विवरण

में बचाया:
ग्रंथसूची विवरण
मुख्य लेखकों: Ponnala, Shashikanth, Gonzales, Junior, Kapadia, Nirav, Navarro, Hernan A., Harding, Wayne W.
स्वरूप: Artigo
भाषा:Inglês
प्रकाशित: 2014
विषय:
ऑनलाइन पहुंच:https://ncbi.nlm.nih.gov/pmc/articles/PMC4022183/
https://ncbi.nlm.nih.gov/pubmed/24630561
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1016/j.bmcl.2014.02.066
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