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C4 phenyl aporphines with selective h5-HT(2B) receptor affinity

A group of aporphine alkaloids related to (±)-nantenine (1) and bearing a C4 phenyl and various C1 or N-substituents, was synthesized and evaluated for affinity to h5-HT receptors. In general, unlike nantenine, the analogues lack affinity for the h5-HT(2A) receptor and other 5-HT receptors but bind...

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Detalhes bibliográficos
Publicado no:Bioorg Med Chem Lett
Main Authors: Kapadia, Nirav, Harding, Wayne W.
Formato: Artigo
Idioma:Inglês
Publicado em: 2015
Assuntos:
Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC4523491/
https://ncbi.nlm.nih.gov/pubmed/26227772
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1016/j.bmcl.2015.07.012
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