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The CYP3A4 intron 6 C>T polymorphism (CYP3A4*22) is associated with reduced CYP3A4 protein level and function in human liver microsomes

Effects of the CYP3A4 intron 6 C>T (CYP3A4*22) polymorphism, which has recently been reported to have a critical role in vivo, were investigated by measuring CYP3A4 protein expression levels and CYP3A4-dependent drug oxidation activities in individual human liver microsomes in vitro. Prior to pro...

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Библиографические подробности
Главные авторы: Okubo, Maho, Murayama, Norie, Shimizu, Makiko, Shimada, Tsutomu, Guengerich, F. Peter, Yamazaki, Hiroshi
Формат: Artigo
Язык:Inglês
Опубликовано: 2013
Предметы:
Online-ссылка:https://ncbi.nlm.nih.gov/pmc/articles/PMC4018728/
https://ncbi.nlm.nih.gov/pubmed/23665933
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