A carregar...

Human Liver Microsomal Cytochrome P450 3A Enzymes Involved in Thalidomide 5-Hydroxylation and Formation of a Glutathione Conjugate

(R)-Thalidomide was oxidized to 5-hydroxythalidomide and 5’-hydroxythalidomide by NADPH-fortified liver microsomes from humans and monkeys. (R)-Thalidomide was hydroxylated more efficiently than (S)-thalidomide. Recombinant human P450s 3A4, 3A5, and 3A7 and monkey P450s 3A8 and 3A5 (co-expressed wit...

ver descrição completa

Na minha lista:
Detalhes bibliográficos
Main Authors: Chowdhury, Goutam, Murayama, Norie, Okada, Yusuke, Uno, Yasuhiro, Shimizu, Makiko, Shibata, Norio, Guengerich, F. Peter, Yamazaki, Hiroshi
Formato: Artigo
Idioma:Inglês
Publicado em: 2010
Assuntos:
Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC3843493/
https://ncbi.nlm.nih.gov/pubmed/20443640
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/tx900367p
Tags: Adicionar Tag
Sem tags, seja o primeiro a adicionar uma tag!