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Role of CYP3A in isoniazid metabolism in vivo

Isoniazid (INH), a first-line drug for tuberculosis control, frequently causes liver injury. Multiple previous reports suggest that CYP3A is involved in INH metabolism, bioactivation and hepatotoxicity, although direct evidence is unavailable. In the current study, wild-type and Cyp3a-null mice were...

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Autors principals: Liu, Ke, Li, Feng, Lu, Jie, Gao, Zhiwei, Klaassen, Curtis D., Ma, Xiaochao
Format: Artigo
Idioma:Inglês
Publicat: 2013
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Accés en línia:https://ncbi.nlm.nih.gov/pmc/articles/PMC4004657/
https://ncbi.nlm.nih.gov/pubmed/24172716
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