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Bedaquiline Metabolism: Enzymes and Novel Metabolites
Bedaquiline is a recently approved drug for the treatment of multidrug-resistant tuberculosis. Adverse cardiac and hepatic drug reactions to bedaquiline have been noted in clinical practice. The current study investigated bedaquiline metabolism in human hepatocytes using a metabolomic approach. Beda...
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Main Authors: | , , , , , , |
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Formato: | Artigo |
Idioma: | Inglês |
Publicado: |
The American Society for Pharmacology and Experimental Therapeutics
2014
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Assuntos: | |
Acceso en liña: | https://ncbi.nlm.nih.gov/pmc/articles/PMC3989786/ https://ncbi.nlm.nih.gov/pubmed/24513655 https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1124/dmd.113.056119 |
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