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Bedaquiline Metabolism: Enzymes and Novel Metabolites

Bedaquiline is a recently approved drug for the treatment of multidrug-resistant tuberculosis. Adverse cardiac and hepatic drug reactions to bedaquiline have been noted in clinical practice. The current study investigated bedaquiline metabolism in human hepatocytes using a metabolomic approach. Beda...

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Main Authors: Liu, Ke, Li, Feng, Lu, Jie, Liu, Shinlan, Dorko, Kenneth, Xie, Wen, Ma, Xiaochao
Formato: Artigo
Idioma:Inglês
Publicado: The American Society for Pharmacology and Experimental Therapeutics 2014
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Acceso en liña:https://ncbi.nlm.nih.gov/pmc/articles/PMC3989786/
https://ncbi.nlm.nih.gov/pubmed/24513655
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1124/dmd.113.056119
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