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Malaria-Infected Mice Are Cured by a Single Low Dose of a New Silylamide Trioxane Plus Mefloquine

Three thermally and hydrolytically stable silylamide trioxanes have been prepared from the natural trioxane artemisinin in only five simple chemical steps and in at least 56% overall yield. Two of these new chemical entities completely cured malaria-infected mice at a single oral dose of only 8 mg/k...

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Detaylı Bibliyografya
Asıl Yazarlar: Woodard, Lauren E., Mott, Bryan T., Singhal, Vandana, Kumar, Nirbhay, Shapiro, Theresa A., Posner, Gary H.
Materyal Türü: Artigo
Dil:Inglês
Baskı/Yayın Bilgisi: Molecular Diversity Preservation International 2009
Konular:
Online Erişim:https://ncbi.nlm.nih.gov/pmc/articles/PMC3978545/
https://ncbi.nlm.nih.gov/pubmed/27713236
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.3390/ph2030228
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