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Conjugation of methotrexate to poly(L-lysine) increases drug transport and overcomes drug resistance in cultured cells

Methotrexate and [(3)H]methotrexate were conjugated through a carbodiimide-catalyzed reaction to a 70,000 molecular weight poly(L-lysine) in molar ratios of approximately 13 to 1. The cellular uptake of labeled conjugate was far in excess of the uptake of free drug in cells that were either proficie...

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Detalles Bibliográficos
Main Authors: Ryser, Hugues J.-P., Shen, Wei-Chiang
Formato: Artigo
Idioma:Inglês
Publicado: 1978
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Acceso en liña:https://ncbi.nlm.nih.gov/pmc/articles/PMC392889/
https://ncbi.nlm.nih.gov/pubmed/279001
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