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Efflux Inhibition with Verapamil Potentiates Bedaquiline in Mycobacterium tuberculosis

Drug efflux is an important resistance mechanism in Mycobacterium tuberculosis. We found that verapamil, an efflux inhibitor, profoundly decreases the MIC of bedaquiline and clofazimine to M. tuberculosis by 8- to 16-fold. This exquisite susceptibility was noted among drug-susceptible and drug-resis...

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Detalhes bibliográficos
Main Authors: Gupta, Shashank, Cohen, Keira A., Winglee, Kathryn, Maiga, Mamoudou, Diarra, Bassirou, Bishai, William R.
Formato: Artigo
Idioma:Inglês
Publicado em: American Society for Microbiology 2014
Assuntos:
Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC3910722/
https://ncbi.nlm.nih.gov/pubmed/24126586
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1128/AAC.01462-13
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