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Autoinhibition of Acetylcholine Binding to Torpedo Electroplax; A Possible Molecular Mechanism for Desensitization

Binding of [(3)H]acetylcholine (measured by equilibrium dialysis) to a particulate preparation of Torpedo electroplax exhibits autoinhibition at concentrations higher than 1 μM. It is suggested that autoinhibition results from acetylcholine binding to regulatory sites on its receptor macromolecules....

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Dades bibliogràfiques
Publicat a:Proc Natl Acad Sci U S A
Autors principals: Eldefrawi, M. E., O'Brien, R. D.
Format: Artigo
Idioma:Inglês
Publicat: National Academy of Sciences 1971
Matèries:
Accés en línia:https://ncbi.nlm.nih.govhttps://pmc.ncbi.nlm.nih.gov/articles/PMC389336/
https://ncbi.nlm.nih.govhttps://pubmed.ncbi.nlm.nih.gov/4332243/
https://ncbi.nlm.nih.govhttps://doi.org/10.1073/pnas.68.9.2006
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