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Autoinhibition of Acetylcholine Binding to Torpedo Electroplax; A Possible Molecular Mechanism for Desensitization
Binding of [(3)H]acetylcholine (measured by equilibrium dialysis) to a particulate preparation of Torpedo electroplax exhibits autoinhibition at concentrations higher than 1 μM. It is suggested that autoinhibition results from acetylcholine binding to regulatory sites on its receptor macromolecules....
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| Главные авторы: | , |
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| Формат: | Artigo |
| Язык: | Inglês |
| Опубликовано: |
1971
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| Предметы: | |
| Online-ссылка: | https://ncbi.nlm.nih.gov/pmc/articles/PMC389336/ https://ncbi.nlm.nih.gov/pubmed/4332243 |
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