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Novel Adamantyl Arotinoids that Inhibit IκB Kinase-α and IκB Kinase-β

A series of analogs of the adamantyl arotinoid (AdAr) chalcone 5 (MX781) having halogenated benzyloxy substituents at C2′ and heterocyclic derivatives replacing the chalcone group were found to inhibit IκBα kinase α (IKKα) and IκBα kinase β (IKKβ) activities. The growth inhibitory activity of some a...

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Autors principals: Lorenzo, Paula, Ortiz, María A., Álvarez, Rosana, Piedrafita, F. Javier, de Lera, Ángel R.
Format: Artigo
Idioma:Inglês
Publicat: 2013
Matèries:
Accés en línia:https://ncbi.nlm.nih.gov/pmc/articles/PMC3892996/
https://ncbi.nlm.nih.gov/pubmed/23653373
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1002/cmdc.201300100
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