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Inhibition of IκB Kinase-β and IκB Kinase-α by Heterocyclic Adamantyl Arotinoids

We recently reported on a series of retinoid-related molecules containing an adamantyl group, a.k.a. adamantyl arotinoids (AdArs), that showed significant cancer cell growth inhibitory activity and activated RXRα (NR2B1) in transient transfection assays while devoid of RAR transactivation capacity....

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Publicat a:Bioorg Med Chem
Autors principals: García-Rodríguez, José, Pérez-Rodríguez, Santiago, Ortiz, María A., Pereira, Raquel, de Lera, Angel R., Piedrafita, F. Javier
Format: Artigo
Idioma:Inglês
Publicat: 2014
Matèries:
Accés en línia:https://ncbi.nlm.nih.gov/pmc/articles/PMC6805150/
https://ncbi.nlm.nih.gov/pubmed/24457093
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1016/j.bmc.2014.01.006
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