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Inhibition of IκB Kinase-β and IκB Kinase-α by Heterocyclic Adamantyl Arotinoids

We recently reported on a series of retinoid-related molecules containing an adamantyl group, a.k.a. adamantyl arotinoids (AdArs), that showed significant cancer cell growth inhibitory activity and activated RXRα (NR2B1) in transient transfection assays while devoid of RAR transactivation capacity....

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Detaylı Bibliyografya
Yayımlandı:Bioorg Med Chem
Asıl Yazarlar: García-Rodríguez, José, Pérez-Rodríguez, Santiago, Ortiz, María A., Pereira, Raquel, de Lera, Angel R., Piedrafita, F. Javier
Materyal Türü: Artigo
Dil:Inglês
Baskı/Yayın Bilgisi: 2014
Konular:
Online Erişim:https://ncbi.nlm.nih.gov/pmc/articles/PMC6805150/
https://ncbi.nlm.nih.gov/pubmed/24457093
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1016/j.bmc.2014.01.006
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