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Pharmacokinetic Assessment of Efflux Transport in Sunitinib Distribution to the Brain

This study quantitatively assessed transport mechanisms that limit the brain distribution of sunitinib and investigated adjuvant strategies to improve its brain delivery for the treatment of glioblastoma multiforme (GBM). Sunitinib has not shown significant activity in GBM clinical trials, despite p...

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Autori principali: Oberoi, Rajneet K., Mittapalli, Rajendar K., Elmquist, William F.
Natura: Artigo
Lingua:Inglês
Pubblicazione: The American Society for Pharmacology and Experimental Therapeutics 2013
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Accesso online:https://ncbi.nlm.nih.gov/pmc/articles/PMC3836310/
https://ncbi.nlm.nih.gov/pubmed/24113148
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1124/jpet.113.208959
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