Wird geladen...

Saturable Active Efflux by P-Glycoprotein and Breast Cancer Resistance Protein at the Blood-Brain Barrier Leads to Nonlinear Distribution of Elacridar to the Central Nervous System

The study objective was to investigate factors that affect the central nervous system (CNS) distribution of elacridar. Elacridar inhibits transport mediated by P-glycoprotein (P-gp) and breast cancer resistance protein (Bcrp) and has been used to study the influence of transporters on brain distribu...

Ausführliche Beschreibung

Gespeichert in:
Bibliographische Detailangaben
Hauptverfasser: Sane, Ramola, Agarwal, Sagar, Mittapalli, Rajendar K., Elmquist, William F.
Format: Artigo
Sprache:Inglês
Veröffentlicht: The American Society for Pharmacology and Experimental Therapeutics 2013
Schlagworte:
Online Zugang:https://ncbi.nlm.nih.gov/pmc/articles/PMC3608446/
https://ncbi.nlm.nih.gov/pubmed/23397054
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1124/jpet.112.199786
Tags: Tag hinzufügen
Keine Tags, Fügen Sie den ersten Tag hinzu!