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Enzymatic Detoxication, Conformational Selection, and the Role of Molten Globule Active Sites

The role of conformational ensembles in enzymatic reactions remains unclear. Discussion concerning “induced fit” versus “conformational selection” has, however, ignored detoxication enzymes, which exhibit catalytic promiscuity. These enzymes dominate drug metabolism and determine drug-drug interacti...

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Bibliografiske detaljer
Main Authors: Honaker, Matthew T., Acchione, Mauro, Zhang, Wei, Mannervik, Bengt, Atkins, William M.
Format: Artigo
Sprog:Inglês
Udgivet: American Society for Biochemistry and Molecular Biology 2013
Fag:
Online adgang:https://ncbi.nlm.nih.gov/pmc/articles/PMC3689999/
https://ncbi.nlm.nih.gov/pubmed/23649628
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1074/jbc.M112.445767
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