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Enzymatic Detoxication, Conformational Selection, and the Role of Molten Globule Active Sites

The role of conformational ensembles in enzymatic reactions remains unclear. Discussion concerning “induced fit” versus “conformational selection” has, however, ignored detoxication enzymes, which exhibit catalytic promiscuity. These enzymes dominate drug metabolism and determine drug-drug interacti...

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שמור ב:
מידע ביבליוגרפי
Main Authors: Honaker, Matthew T., Acchione, Mauro, Zhang, Wei, Mannervik, Bengt, Atkins, William M.
פורמט: Artigo
שפה:Inglês
יצא לאור: American Society for Biochemistry and Molecular Biology 2013
נושאים:
גישה מקוונת:https://ncbi.nlm.nih.gov/pmc/articles/PMC3689999/
https://ncbi.nlm.nih.gov/pubmed/23649628
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1074/jbc.M112.445767
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