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PARP and CHK inhibitors interact to cause DNA damage and cell death in mammary carcinoma cells

The present studies examined viability and DNA damage levels in mammary carcinoma cells following PARP1 and CHK1 inhibitor drug combination exposure. PARP1 inhibitors [AZD2281 ; ABT888 ; NU1025 ; AG014699] interacted with CHK1 inhibitors [UCN-01 ; AZD7762 ; LY2603618] to kill mammary carcinoma cells...

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Détails bibliographiques
Auteurs principaux: Booth, Laurence, Cruickshanks, Nichola, Ridder, Thomas, Dai, Yun, Grant, Steven, Dent, Paul
Format: Artigo
Langue:Inglês
Publié: Landes Bioscience 2013
Sujets:
Accès en ligne:https://ncbi.nlm.nih.gov/pmc/articles/PMC3672190/
https://ncbi.nlm.nih.gov/pubmed/23917378
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.4161/cbt.24424
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