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An X-ray Snapshot of the Mechanism of Inactivation of Human Neutrophil Elastase by 1, 2, 5 –Thiadiazolidin-3-one 1, 1 Dioxide Derivatives

The mechanism of action of a general class of mechanism-based inhibitors of serine proteases, including human neutrophil elastase (HNE), has been elucidated by determining the X-ray crystal structure of an enzyme-inhibitor complex. The captured intermediate indicates that processing of inhibitor (I)...

Täydet tiedot

Tallennettuna:
Bibliografiset tiedot
Päätekijät: Huang, Weijun, Yamamoto, Yasufumi, Li, Yi, Dou, Dengfeng, Alliston, Kevin R., Hanzlik, Robert P., Williams, Todd D., Groutas, William C.
Aineistotyyppi: Artigo
Kieli:Inglês
Julkaistu: 2008
Aiheet:
Linkit:https://ncbi.nlm.nih.gov/pmc/articles/PMC3623276/
https://ncbi.nlm.nih.gov/pubmed/18318470
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/jm700966p
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