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Substituted phenyl groups improve the pharmacokinetic profile and anti-inflammatory effect of urea-based soluble epoxide hydrolase inhibitors in murine models

Soluble epoxide hydrolase inhibitors (sEHIs) are anti-inflammatory, analgesic, anti-hypertensive, cardio- and renal-protective in multiple animal models. However, the earlier adamantyl-containing urea-based inhibitors are rapidly metabolized. Therefore, new potent inhibitors with the adamantyl group...

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Détails bibliographiques
Auteurs principaux: Liu, Jun-Yan, Lin, Yan-Ping, Qiu, Hong, Morisseau, Christophe, Rose, Tristan E., Hwang, Sung Hee, Chiamvimonvat, Nipavan, Hammock, Bruce D.
Format: Artigo
Langue:Inglês
Publié: 2013
Sujets:
Accès en ligne:https://ncbi.nlm.nih.gov/pmc/articles/PMC3596469/
https://ncbi.nlm.nih.gov/pubmed/23291046
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1016/j.ejps.2012.12.013
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