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Substituent Effects on Desferrithiocin and Desferrithiocin Analogue Iron Clearing and Toxicity Profiles

Desferrithiocin (DFT, 1) is a very efficient iron chelator when given orally. However, it is severely nephrotoxic. Structure-activity studies with 1 demonstrated that removal of the aromatic nitrogen to provide desazadesferrithiocin (DADFT, 2) and introduction of either a hydroxyl group or a polyeth...

Ausführliche Beschreibung

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Bibliographische Detailangaben
Hauptverfasser: Bergeron, Raymond J., Wiegand, Jan, Bharti, Neelam, McManis, James S.
Format: Artigo
Sprache:Inglês
Veröffentlicht: 2012
Schlagworte:
Online Zugang:https://ncbi.nlm.nih.gov/pmc/articles/PMC3583384/
https://ncbi.nlm.nih.gov/pubmed/22889170
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/jm300509y
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