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Methadone metabolism and clearance are induced by nelfinavir despite inhibition of cytochrome P4503A (CYP3A) activity

BACKGROUND: Methadone plasma concentrations are decreased by nelfinavir. Methadone clearance and the drug interactions have been attributed to CYP3A4, but actual mechanisms of methadone clearance and the nelfinavir interaction are unknown. We assessed nelfinavir effects on methadone pharmacokinetics...

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Autores principales: Kharasch, Evan D., Walker, Alysa, Whittington, Dale, Hoffer, Christine, Bedynek, Pamela Sheffels
Formato: Artigo
Lenguaje:Inglês
Publicado: 2009
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Acceso en línea:https://ncbi.nlm.nih.gov/pmc/articles/PMC3582041/
https://ncbi.nlm.nih.gov/pubmed/19232844
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1016/j.drugalcdep.2008.12.009
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