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Methadone Pharmacokinetics are Independent of Cytochrome P4503A (CYP3A) Activity and Gastrointestinal Drug Transport: Insights from Methadone Interactions with Ritonavir/Indinavir

BACKGROUND: Methadone clearance is highly variable and drug interactions are problematic. Both have been attributed to CYP3A, but actual mechanisms are unknown. Drug interactions can provide such mechanistic information. Ritonavir/indinavir, one of the earliest protease inhibitor combinations, may i...

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Autori principali: Kharasch, Evan D., Hoffer, Christine, Whittington, Dale, Walker, Alysa, Bedynek, Pamela Sheffels
Natura: Artigo
Lingua:Inglês
Pubblicazione: 2009
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Accesso online:https://ncbi.nlm.nih.gov/pmc/articles/PMC3111241/
https://ncbi.nlm.nih.gov/pubmed/19225389
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1097/ALN.0b013e3181986a9a
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