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Antitumor activity of a pyrrole-imidazole polyamide

Many cancer therapeutics target DNA and exert cytotoxicity through the induction of DNA damage and inhibition of transcription. We report that a DNA minor groove binding hairpin pyrrole-imidazole (Py-Im) polyamide interferes with RNA polymerase II (RNAP2) activity in cell culture. Polyamide treatmen...

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Détails bibliographiques
Auteurs principaux: Yang, Fei, Nickols, Nicholas G., Li, Benjamin C., Marinov, Georgi K., Said, Jonathan W., Dervan, Peter B.
Format: Artigo
Langue:Inglês
Publié: National Academy of Sciences 2013
Sujets:
Accès en ligne:https://ncbi.nlm.nih.gov/pmc/articles/PMC3562772/
https://ncbi.nlm.nih.gov/pubmed/23319609
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1073/pnas.1222035110
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