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Validation of the proteasome as a therapeutic target in Plasmodium using an epoxyketone inhibitor with parasite-specific toxicity

The Plasmodium proteasome has been suggested to be a potential anti-malarial drug target, however toxicity of inhibitors has prevented validation of this enzyme in vivo. We report here a screen of a library of 670 analogs of the recently FDA approved inhibitor, carfilzomib, to identify compounds tha...

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Detalhes bibliográficos
Main Authors: Li, Hao, Ponder, Elizabeth L., Verdoes, Martijn, Asbjornsdottir, Kristijana H., Deu, Edgar, Edgington, Laura E., Lee, Jeong Tae, Kirk, Christopher J., Demo, Susan D., Williamson, Kim C., Bogyo, Matthew
Formato: Artigo
Idioma:Inglês
Publicado em: 2012
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Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC3529830/
https://ncbi.nlm.nih.gov/pubmed/23142757
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1016/j.chembiol.2012.09.019
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