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Dynamics connect substrate recognition to catalysis in protein kinase A

Atomic resolution studies of protein kinases have traditionally been carried out in the inhibitory state, limiting our current knowledge on the mechanisms of substrate recognition and catalysis. Using NMR, x-ray crystallography, and thermodynamic measurements we analyzed the substrate recognition pr...

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Autores principales: Masterson, Larry R., Cheng, Cecilia, Yu, Tao, Tonelli, Marco, Kornev, Alexandr, Taylor, Susan S., Veglia, Gianluigi
Formato: Artigo
Lenguaje:Inglês
Publicado: 2010
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Acceso en línea:https://ncbi.nlm.nih.gov/pmc/articles/PMC3487389/
https://ncbi.nlm.nih.gov/pubmed/20890288
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1038/nchembio.452
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