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Fragment screening of cyclin G-associated kinase by weak affinity chromatography

Fragment-based drug discovery (FBDD) has become a new strategy for drug discovery where lead compounds are evolved from small molecules. These fragments form low affinity interactions (dissociation constant (K(D)) = mM − μM) with protein targets, which require fragment screening methods of sufficien...

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Autors principals: Meiby, Elinor, Knapp, Stefan, Elkins, Jonathan M., Ohlson, Sten
Format: Artigo
Idioma:Inglês
Publicat: Springer-Verlag 2012
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Accés en línia:https://ncbi.nlm.nih.gov/pmc/articles/PMC3475971/
https://ncbi.nlm.nih.gov/pubmed/22918538
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1007/s00216-012-6335-6
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