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Towards the Development of an In vivo Chemical Probe for Cyclin G Associated Kinase (GAK)
SGC-GAK-1 (<b>1</b>) is a potent, selective, cell-active chemical probe for cyclin G-associated kinase (GAK). However, <b>1</b> was rapidly metabolized in mouse liver microsomes by cytochrome P450-mediated oxidation, displaying rapid clearance in liver microsomes and in mice,...
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| Autors principals: | , , , , , , , , , |
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| Format: | Artigo |
| Idioma: | Inglês |
| Publicat: |
MDPI AG
2019-11-01
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| Col·lecció: | Molecules |
| Matèries: | |
| Accés en línia: | https://www.mdpi.com/1420-3049/24/22/4016 |
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