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Inhibition of protease-activated receptor 1 ameliorates intestinal radiation mucositis in a preclinical rat model

SUMMARY: Direct inhibition of thrombin has a beneficial effect on intestinal radiation toxicity. A small molecule inhibitor of protease-activated receptor 1 (PAR1), the most relevant receptor for thrombin, was administered to rats undergoing localized, fractionated irradiation of a segment of small...

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Detalhes bibliográficos
Main Authors: Wang, Junru, Kulkarni, Ashwini, Chintala, Madhu, Fink, Louis M., Hauer-Jensen, Martin
Formato: Artigo
Idioma:Inglês
Publicado em: 2012
Assuntos:
Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC3462888/
https://ncbi.nlm.nih.gov/pubmed/22580123
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1016/j.ijrobp.2012.02.007
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