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The genesis of Zelboraf: Targeting mutant B-Raf in melanoma

The protein kinase B-Raf is a critical component of the Ras/MAPK signaling pathway. An oncogenic B-Raf mutation that constitutively activates the kinase was identified in z50% of melanoma patients and in other cancers. A structure-guided drug discovery approach enabled the development of Zelboraf, a...

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Autori principali: Davis, Matthew J., Schlessinger, Joseph
Natura: Artigo
Lingua:Inglês
Pubblicazione: The Rockefeller University Press 2012
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Accesso online:https://ncbi.nlm.nih.gov/pmc/articles/PMC3461519/
https://ncbi.nlm.nih.gov/pubmed/23027900
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1083/jcb.201205167
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