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A FUNCTIONAL SCREENING OF ADENOSINE ANALOGUES AT THE ADENOSINE A(2B) RECEPTOR: A SEARCH FOR POTENT AGONISTS
Various adenosine analogues were tested at the adenosine A(2B) receptor. Agonist potencies were determined by measuring the cyclic AMP production in Chinese Hamster Ovary cells expressing human A(2B) receptors. 5′-N-Substituted carboxamidoadenosines were most potent. 5′-N-Ethylcarboxamidoadenosine (...
Αποθηκεύτηκε σε:
| Κύριοι συγγραφείς: | , , , , , , |
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| Μορφή: | Artigo |
| Γλώσσα: | Inglês |
| Έκδοση: |
1998
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| Θέματα: | |
| Διαθέσιμο Online: | https://ncbi.nlm.nih.gov/pmc/articles/PMC3459057/ https://ncbi.nlm.nih.gov/pubmed/9708319 https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1080/07328319808004215 |
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