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Profiling the Dynamic Interfaces of Fluorinated Transcription Complexes for Ligand Discovery and Characterization

The conformationally dynamic binding surfaces of transcription complexes present a particular challenge for ligand discovery and characterization. In the case of the KIX domain of the master coactivator CBP/p300, few small molecules have been reported that target its two allosterically regulated bin...

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Autores principales: Pomerantz, William C., Wang, Ningkun, Lipinski, Ashley K., Wang, Rurun, Cierpicki, Tomasz, Mapp, Anna K.
Formato: Artigo
Lenguaje:Inglês
Publicado: 2012
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Acceso en línea:https://ncbi.nlm.nih.gov/pmc/articles/PMC3423543/
https://ncbi.nlm.nih.gov/pubmed/22725662
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/cb3002733
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