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Lysosomal delivery of a lipophilic gemcitabine prodrug using novel acid-sensitive micelles improved its antitumor activity

Stimulus-sensitive micelles are attractive anticancer drug delivery systems. Herein we reported a novel strategy to engineer acid-sensitive micelles using a amphiphilic material synthesized by directly conjugating the hydrophilic polyethylene glycol (PEG) with a hydrophobic stearic acid derivative (...

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Autors principals: Zhu, Saijie, Lansakara-P, Dharmika S.P., Li, Xinran, Cui, Zhengrong
Format: Artigo
Idioma:Inglês
Publicat: 2012
Matèries:
Accés en línia:https://ncbi.nlm.nih.gov/pmc/articles/PMC3419313/
https://ncbi.nlm.nih.gov/pubmed/22471294
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/bc2005945
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