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Plasma Pharmacokinetics and Tissue Disposition of Novel Dextran- Methylprednisolone Conjugates with Peptide Linkers in Rats

The plasma and tissue disposition of two novel dextran prodrugs of methylprednisolone (MP) containing one (DMP-1) or five (DMP-5) amino acids as linkers were studied in rats. Single 5-mg/kg doses (MP equivalent) of each prodrug or MP were administered intravenously, and blood and tissue samples were...

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Autors principals: Penugonda, Suman, Agarwal, Hitesh K., Parang, Keykavous, Mehvar, Reza
Format: Artigo
Idioma:Inglês
Publicat: 2010
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Accés en línia:https://ncbi.nlm.nih.gov/pmc/articles/PMC3415712/
https://ncbi.nlm.nih.gov/pubmed/19780131
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1002/jps.21934
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