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Ranolazine Decreases Mechanosensitivity of the Voltage-Gated Sodium Ion Channel Na(V)1.5: A Novel Mechanism of Drug Action

BACKGROUND: Na(V)1.5 is a mechanosensitive voltage gated sodium-selective ion channel responsible for the depolarizing current and maintenance of the action potential plateau in the heart. Ranolazine is a Na(V)1.5 antagonist with anti-anginal and anti-arrhythmic properties. METHODS AND RESULTS: Mech...

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Main Authors: Beyder, Arthur, Strege, Peter R., Reyes, Santiago, Bernard, Cheryl E., Terzic, Andre, Makielski, Jonathan, Ackerman, Michael J., Farrugia, Gianrico
Formato: Artigo
Idioma:Inglês
Publicado: 2012
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Acceso en liña:https://ncbi.nlm.nih.gov/pmc/articles/PMC3392778/
https://ncbi.nlm.nih.gov/pubmed/22565935
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1161/CIRCULATIONAHA.112.094714
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