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Brain Distribution of Cediranib Is Limited by Active Efflux at the Blood-Brain Barrier

Cediranib is an orally active tyrosine kinase inhibitor that targets the vascular endothelial growth factor receptor family. Because of its potent antiangiogenic and antitumor activities, cediranib has been evaluated for therapy in glioma, a primary brain tumor. This study investigated the influence...

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Autori principali: Wang, Tianli, Agarwal, Sagar, Elmquist, William F.
Natura: Artigo
Lingua:Inglês
Pubblicazione: The American Society for Pharmacology and Experimental Therapeutics 2012
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Accesso online:https://ncbi.nlm.nih.gov/pmc/articles/PMC3336816/
https://ncbi.nlm.nih.gov/pubmed/22323823
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1124/jpet.111.190488
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