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P-glycoprotein-Based Loperamide-Cyclosporine Drug Interaction at the Rat Blood-Brain Barrier: Prediction from In Vitro Studies and Extrapolation to Humans

We have shown that the rat can quantitatively predict the verapamil-cyclopsorine A (CsA) drug-drug interaction (DDI) at the human blood-brain barrier (BBB). In addition, the potency (EC(50)) of CsA to inhibit rat BBB P-gp can be predicted from in vitro studies in MDRI-transfected cells. To assess if...

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Bibliografski detalji
Glavni autori: Hsiao, Peng, Unadkat, Jashvant D.
Format: Artigo
Jezik:Inglês
Izdano: 2012
Teme:
Online pristup:https://ncbi.nlm.nih.gov/pmc/articles/PMC3307806/
https://ncbi.nlm.nih.gov/pubmed/22316009
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/mp200563a
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