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Targeting Diverse Signaling Interaction Sites Allows the Rapid Generation of Bivalent Kinase Inhibitors

The identification of potent and selective modulators of protein kinase function remains a challenge and new strategies are needed for generating these useful ligands. Here, we describe the generation of bivalent inhibitors of three unrelated protein kinases: the CAMK family kinase Pim1, the mitogen...

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Hlavní autoři: Hill, Zachary B., Perera, B. Gayani K., Andrews, Simeon S., Maly, Dustin J.
Médium: Artigo
Jazyk:Inglês
Vydáno: 2011
Témata:
On-line přístup:https://ncbi.nlm.nih.gov/pmc/articles/PMC3306478/
https://ncbi.nlm.nih.gov/pubmed/22148755
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/cb200387g
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