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Rapid profiling of protein kinase inhibitors by quantitative proteomics

The ability to determine structure-activity relationships (SAR) and identify cellular targets from cell lysates and tissues is of great utility for kinase inhibitor drug discovery. We describe a streamlined mass spectrometry-based chemoproteomics workflow to examine the SAR and target profiles of a...

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Détails bibliographiques
Auteurs principaux: Golkowski, Martin, Brigham, Jennifer L., Perera, Gayani K., Romano, Guillermo E., Maly, Dustin J., Ong, Shao-En
Format: Artigo
Langue:Inglês
Publié: 2014
Sujets:
Accès en ligne:https://ncbi.nlm.nih.gov/pmc/articles/PMC3955727/
https://ncbi.nlm.nih.gov/pubmed/24648882
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1039/C3MD00315A
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