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Advances in the clinical development of heat shock protein 90 (Hsp90) inhibitors in cancers

Hsp90 is an ATP dependent molecular chaperone protein which integrates multiple oncogenic pathways. As such, Hsp90 inhibition is a promising anti-cancer strategy. Several inhibitors that act on Hsp90 by binding to its N-terminal ATP pocket have entered clinical evaluation. Robust pre-clinical data s...

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Bibliografski detalji
Glavni autori: Jhaveri, Komal, Taldone, Tony, Modi, Shanu, Chiosis, Gabriela
Format: Artigo
Jezik:Inglês
Izdano: 2011
Teme:
Online pristup:https://ncbi.nlm.nih.gov/pmc/articles/PMC3288123/
https://ncbi.nlm.nih.gov/pubmed/22062686
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1016/j.bbamcr.2011.10.008
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