Загрузка...

Identification of novel SAR properties of the Jak2 small molecule inhibitor G6: significance of the para-hydroxyl orientation

In this study, we analyzed the structure activity relationship properties of the small molecule Jak2 inhibitor G6. We synthesized a set of derivatives containing the native para-hydroxyl structure or an alternative meta-hydroxyl structure and examined their Jak2 inhibitory properties. We found that...

Полное описание

Сохранить в:
Библиографические подробности
Главные авторы: Baskin, Rebekah, Gali, Meghanath, Park, Sung O., Zhao, Zhizhuang Joe, Keserű, György M., Bisht, Kirpal S., Sayeski, Peter P.
Формат: Artigo
Язык:Inglês
Опубликовано: 2011
Предметы:
Online-ссылка:https://ncbi.nlm.nih.gov/pmc/articles/PMC3267892/
https://ncbi.nlm.nih.gov/pubmed/22227213
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1016/j.bmcl.2011.12.042
Метки: Добавить метку
Нет меток, Требуется 1-ая метка записи!