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Molecular Determinants of Pentamidine-Induced hERG Trafficking Inhibition

Pentamidine is an antiprotozoal compound that clinically causes acquired long QT syndrome (acLQTS), which is associated with prolonged QT intervals, tachycardias, and sudden cardiac arrest. Pentamidine delays terminal repolarization in human heart by acutely blocking cardiac inward rectifier current...

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Main Authors: Dennis, Adrienne T., Wang, Lu, Wan, Hanlin, Nassal, Drew, Deschenes, Isabelle, Ficker, Eckhard
Formato: Artigo
Idioma:Inglês
Publicado: The American Society for Pharmacology and Experimental Therapeutics 2012
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Acceso en liña:https://ncbi.nlm.nih.gov/pmc/articles/PMC3263949/
https://ncbi.nlm.nih.gov/pubmed/22046004
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1124/mol.111.075135
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